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Next-Gen Kinase Inhibitors(次世代激酶抑制剂学会) | 2011年6月6-8日, 美国剑桥



主题重点

Arrow选择性的设计、筛选、评估

Arrow变构激酶抑制剂的特定与分析

Arrow共享结合阻碍

Arrow中枢神经系适应的激酶:大课题

Arrow炎症与自体免疫—主要计画

Arrow癌的激酶—PI3、mTOR、cMet等

Arrow追求新的激酶标的

ArrowDMPK、Tox的筛选与监测

Arrow计算机手法的进化

Arrow抵抗性—将来的课题


Click here for the preliminary agenda


著名的学术相关人员

Mark Ashwell, ArQule Inc

Peter Brandt, Beactica AB

Dirksen Bussiere, Novartis Vaccines & Diagnostics Inc.

Jean Cui, Pfizer, Inc.

Greg Cuny, Brigham & Women’s Hospital

David C. Dalgarno, ARIAD Pharmaceuticals Inc.

David H. Drewry, GlaxoSmithKline

Isabelle Dussault, Amgen

Doriano M. Fabbro, Novartis Institutes for BioMedical Research

Daniel Goldberg, Boehringer-Ingelheim Pharmaceuticals

Andrew C. Good, Genzyme Corp

John D. Haley, OSI Pharmaceuticals

Ronald Knegtel, Vertex Pharmaceuticals (Europe) Ltd.

Ravi G. Kurumbail, Pfizer, Inc.

Chris Liang, Xcovery, LLC

Carol MacKintosh, University of Dundee

Yibing Shan, D. E. Shaw Research

Juswinder Singh, Avila Therapeutics, Inc.

Rajinder Singh, Rigel Pharmaceuticals Inc.

Eli Wallace, Array BioPharma

Neil Wishart, Abbott

Paul Yu, Massachusetts General Hospital



特别专题讨论会:

I. 次世代激酶 ―
选择性与现状

II. 设计基本构造的激酶抑制剂

由对激酶研究有10年以上贡献的精选专题讨论小组参加者们发表。


6月6日 Pre-conference 短期课程(半日)

The Art and Science of Kinases -
What you Need to Know
(激酶的艺术价值与科学—应事先知道的事)

Kent Stewart, Ph.D. Research Fellow, Abbott


 

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